Papers

M. Larhed, C. Moberg, and A. Hallberg:

Microwave-accelerated homogeneous catalysis in organic chemistry.

Accounts of Chemical Research, 35, 717-727 (2002).

 

P. Johannesson, G. Lindeberg, A. Johansson, G. V. Nikiforovich, A. Gogoll, B. Synnergren, M. Le Greves, F. Nyberg, A. Karlen, and A. Hallberg:

Vinyl sulfide cyclized analogues of angiotensin II with high affinity and full agonist activity at the AT(1) receptor.

Journal of Medicinal Chemistry, 45, 1767-1777 (2002).

 

W. Schaal, A. Karlsson, G. Ahlsen, J. Lindberg, H. O. Andersson, U. H. Danielson, B. Classon, T. Unge, B. Samuelsson, J. Hulten, A. Hallberg, and A. Karlen:

Synthesis and comparative molecular field analysis (CoMFA) of symmetric and nonsymmetric cyclic sulfamide HIV-1 protease inhibitors.

Journal of Medicinal Chemistry, 45, 752-752 (2002).

 

P. Nilsson, H. Gold, M. Larhed, and A. Hallberg: Microwave-assisted enantioselective Heck reactions:

Expediting high reaction speed and preparative convenience.

Synthesis, 11, 1611-1614 (2002).

 

P. O. Markgren, W. Schaal, M. Hamalainen, A. Karlen, A. Hallberg, B. Samuelsson, and U. H. Danielson:

Relationships between structure and interaction kinetics for HIV-1 protease inhibitors.

Journal of Medicinal Chemistry, 45, 5430-5439 (2002).

 

A. Bengtson, A. Hallberg, and M. Larhed:

Fast synthesis of aryl triflates with controlled microwave heating.

Organic Letters, 4, 1231-1233 (2002).

 

N. F. K. Kaiser, A. Hallberg, and M. Larhed:

In situ generation of carbon monoxide from solid molybdenum hexacarbonyl. A convenient and fast route to palladium- catalyzed carbonylation reactions.

Journal of Combinatorial Chemistry, 4, 109-111 (2002).

 

Y. Q. Wan, M. Alterman, M. Larhed, and A. Hallberg:

Dimethylformamide as a carbon monoxide source in fast palladium-catalyzed aminocarbonylations of aryl bromides.

Journal of Organic Chemistry, 67, 6232-6235 (2002).

 

Y. Q. Wan, M. Alterman, and A. Hallberg:

Palladium-catalyzed amination of aryl bromides using temperature-controlled microwave heating.

Synthesis-Stuttgart, , 1597-1600 (2002).

 

A. Bengtson, M. Larhed, and A. Hallberg:

Protected indanones by a Heck-Aldol annulation reaction.

Journal of Organic Chemistry, 67, 5854-5856 (2002).

 

M. Erdelyi, V. Langer, A. Karlen, and A. Gogoll:

Insight into beta-hairpin stability: a structural and thermodynamic study of diastereomeric beta-hairpin mimetics.

New Journal of Chemistry, 26, 834-843 (2002).

 

K. S. A. Vallin, P. Emilsson, M. Larhed, and A. Hallberg:

High-speed Heck reactions in ionic liquid with controlled microwave heating.

Journal of Organic Chemistry, 67, 6243-6246 (2002).

 

L. Afzelius, C. M. Masimirembwa, A. Karlen, T. B. Andersson, and I. Zamora:

Discriminant and quantitative PLS analysis of competitive CYP2C9 inhibitors versus non-inhibitors using alignment independent GRIND descriptors.

Journal of Computer-Aided Molecular Design, 16, 443-458 (2002).

 

J. Gabrielsson, N. O. Lindberg, and T. Lundstedt:

Multivariate methods in pharmaceutical applications.

Journal of Chemometrics, 16, 141-160 (2002).

 

M. Lapinsh, A. Gutcaits, P. Prusis, C. Post, T. Lundstedt, and J. E. S. Wikberg:

Classification of G-protein coupled receptors by alignment- independent extraction of principal chemical properties of primary amino acid sequences.

Protein Science, 11, 795-805 (2002).

 

S. L. Payne, A. M. Johansson, and P. G. Strange:

Mechanisms of ligand binding and efficacy at the human D- 2(short) dopamine receptor.

Journal of Neurochemistry, 82, 1106-1117 (2002).

 

A. Johansson, A. Poliakov, E. Akerblom, G. Lindeberg, S. Winwarter, B. Samuelsson, U. H. Danielson, and A. Hallberg:

Tetrapeptides as potent protease inhibitors of hepatitis C virus full-length NS3 (protease-helicase/NTPase).

Bioorganic & Medicinal Chemistry, 10, 3915-3922 (2002).

 

M. Dambrova, M. Veveris, H. Cirule, O. Pugovichs, C. Post, T. Lundstedt, L. Kalvinsh, A. Skottner, and J. E. S. Wikberg:

The novel guanidine ME10092 protects the heart during ischemia- reperfusion.

European Journal of Pharmacology, 445, 105-113 (2002).

 

M. Lapinsh, P. Prusis, T. Lundstedt, and J. E. S. Wikberg:

Proteochemometrics modeling of the interaction of amine G- protein coupled receptors with a diverse set of ligands.

Molecular Pharmacology, 61, 1465-1475 (2002).

 

P. M. Andersson and T. Lundstedt:

Hierarchical experimental design exemplified by QSAR evaluation of a chemical library directed towards the melanocortin 4 receptor.

Journal of Chemometrics, 16, 490-496 (2002).

 

S. H. L. de Villiers, N. Lindblom, G. Kalayanov, S. Gordon, A. Malmerfelt, A. M. Johansson, and T. H. Svensson:

Active immunization against nicotine suppresses nicotine- induced dopamine release in the rat nucleus accumbens shell.

Respiration, 69, 247-253 (2002).

 

M. Almeida, A. Boman, and T. Lundstedt:

Synthesis of N-(2-chloro-3,4- dimethoxybenzylideneamino)guanidinium acetate [alpha-C-14].

Journal of Labelled Compounds & Radiopharmaceuticals, 45, 371-377 (2002).

 

N. O. Lindberg, A. Berdal, G. Enstad, E. Seifert, and T. Lundstedt:

Investigation of flow properties of powders by means of a uniaxial tester, in relation to direct tablet compression.

Drug Development and Industrial Pharmacy, 28, 15-28 (2002).

 

N. Lindblom, S. H. L. de Villiers, G. Kalayanov, S. Gordon, A. M. Johansson, and T. H. Svensson:

Active immunization against nicotine prevents reinstatement of nicotine-seeking behavior in rats.

Respiration, 69, 254-260 (2002).