Papers

A. Arefalk, M. Larhed and A. Hallberg:

Masked 3-Aminoindan-1-ones by a Palladium-Catalyzed Three-Component Annulation Reaction.

J. Org. Chem., 70 (2005) 938-942

 

A. Ax, W. Schaal, L. Vrang, B. Samuelsson,, A. Hallberg, A. Karlén:

Cyclic sulfamide HIV-1 protease inhibitors, with side chains spanning from P2/P2´to P1/P1'.

Bioorg Med Chem 13 (2005) 755-764.

 

A. Svennebring, N. Garg, P. Nilsson, A. Hallberg, M. Larhed:

An one-pot isomerization-arylation of 2,3-epoxycyclohexanone under controlled microwave heating.

J Org Chem 70 (2005) 4720-4725.

 

U. Rosenström, C. Sköld, B. Plouffe, H. Beaudry, G. Lindeberg, M. Botros, F. Nyberg, G. Wolf, A. Karlén, N. Gallo-Payet, A. Hallberg:

New selective AT2 receptor ligands encompassing a γ-turn mimetic replacing the amino acid residues 4-5 of angiotensin II act as agonists.

J Med Chem 48 (2005) 4009-4024.

 

X. Wu, P. Nilsson and M. Larhed:

Microwave-Enhanced Carbonylative Generation of Indanones and 3-Acylaminoindanones.

J. Org. Chem., 70 (2005) 346-349

 

P. O. Johansson, J. Lindberg, M. J. Blackman, I. Kvarnström, L. Vrang, E. Hamelink, A. Hallberg, Å. Rosenquist, B. Samuelsson:

Design and synthesis of potent inhibitors of plasmepsin I and II: X-ray crystal structure of inhibitor in complex with plasmepsin II.

J Med Chem, 48 (2005) 4400-4409.

 

D. Muthas, D. Nöteberg, Y. A. Sabnis, E. Hamelink, L. Vrang, B. Samuelsson, A. Karlén, A. Hallberg:

Synthesis, biological evaluation and modeling studies of inhibitors aimed at the malarial proteases plasmepsin I and II.

Bioorg Med Chem, 13 (2005) 5371-5390.

 

J. Wannberg, N.-F. Kaiser, L. Vrang, B. Samuelsson, M. Larhed, A. Hallberg:

High-speed synthesis of potent C2-symmetric HIV-1 protease inhibitors by in-situ aminocarbonylations.

J Comp Chem, 7 (2005) 611-617.

 

K. Ersmark, M. Nervall, E. Hamelink, L. K. Janka, J. C. Clemente, B. M. Dunn, M. J. Blackman, B. Samuelsson, J. Åqvist, A. Hallberg:

Synthesis of malarial plasmepsin inhibitors and prediction of binding modes by molecular dynamics simulations.

J Med Chem, 48 (2005) 6090-6106.

 

J. K. Ekegren, T. Unge, M. Z. Safa, H. Wallberg, B. Samuelsson, A. Hallberg:

A new class of HIV-1 protease inhibitors containing a tertiary alcohol in the transition-state mimicking scaffold.

J Med Chem, 48 (2005) 8098-8102.

 

J. Georgsson, C. Sköld, B. Plouffe, G. Lindeberg, M. Botros, M. Larhed, F. Nyberg, N. Gallo-Payet, A. Karlén, A. Hallberg:

Angiotensin II pseudopeptides containing 1,3,5-trisubstituted benzene scaffolds with high AT2 receptor affinity.

J Med Chem, 48 (2005) 6620-6631.

 

J. Wannberg, D. Dallinger, C. O. Kappe, and M. Larhed:

Novel Microwave-Enhanced and Metal-Catalyzed Functionalizations of the 4-Aryl-Dihydropyrimidone Template.

J. Comb. Chem., 7 (2005) 574-583

 

P.-A. Enquist, J. Edin, P. Nilsson and M. Larhed:

Super Fast Cobalt Carbonyl-Mediated Synthesis of Urea Compounds.

Tetrahedron Lett., 46 (2005) 3335-3339

 

X. Wu, R. Rönn, T. Gossas and M. Larhed:

Easy-to-Execute Carbonylations: Microwave Synthesis of Acyl Sulfonamides using Mo(CO)₆ as a Solid Carbon Monoxide Source.

J. Org. Chem, 70 (2005) 3094-3098

 

H. Gold, M. Larhed and P. Nilsson:

Microwave Irradiation as a High-Speed Tool for Activation of Sluggish Aryl Chlorides in Grignard Reactions.

Synlett, (2005) 1596-1600

 

X. Wu and Mats Larhed:

Microwave-Enhanced Aminocarbonylations in Water.

Org. Lett., 7 (2005) 3327-3329.