2009

Sorin Srbu — Wed, 14 Jan 2009 08:13:25 GMT

Research papers

A. Trejos, A. Fardost, S. Yahiaoui, M. Larhed*:

Chelation-controlled palladium(II)-catalyzed oxidative coupling reactions with arylboronic acids: A new Heck/Suzuki domino diarylation reaction.

Chem. Commun. Accepted

M. Andaloussi, J. Lindh, J. Sävmarker, P. J. R. Sjöberg, M. Larhed*:

Base-Free Microwave-Promoted Palladium(II)-Catalyzed C-P Bond Formation Using Arylboronic Acids or Aryltrifluoroborates.

Chem. Eur. J., Accepted

A. K. Mahalingam, L. Axelsson, J. K. Ekegren, J. Wannberg, J. Kihlström, T. Unge, H. Wallberg, B. Samuelsson, M. Larhed*, A. Hallberg:

HIV-1 Protease Inhibitors with a Transition-State Mimic Comprising a Tertiary Alcohol: Improved Antiviral Activity in Cells.

Submitted

F. Russo, J. Sävmarker, M. Jacobsson, M. Larhed*:

Synthesis and evaluation of a new class of tertiary alcohol based BACE-1 inhibitors.

Tetrahedron, 65 (2009), 10047-10059.

M. T. Nilsson, W. W. Krajewski, S. Yellagunda, S. Prabhumurthy, G. N. Chamarahally, C. Siddamadappa, B. R. Srinivasa, S. Yahiaoui, M. Larhed, A. Karlén, T. A. Jones, S. L. Mowbray*:

Structural Basis For The Inhibition Of Mycobacterium Tuberculosis Glutamine Synthetase By Novel ATP-Competitive

Inhibitors.

J. Mol. Biol., 393 (2009), 504-513.

J. Lindh, J. Sävmarker, P. Nilsson, P. J. R. Sjöberg, Mats Larhed*:

Synthesis of Styrenes by Direct Palladium(II)-Catalyzed Vinylation of Arylboronic Acids and Aryltrifluoroborates Using Vinyl Acetate.

Chem. Eur. J., 15 (2009), 4630-4636.

J. Lindh, Mats Larhed*:

Microwave-Assisted Palladium(II)-Catalyzed Heck Reactions with Arylboronic Acids.

Chemistry Today, 27 (2009), 2, 11-14.

J. Gising, P. Örtqvist, A. Sandström, Mats Larhed*:

A Straightforward Microwave Method for Rapid Synthesis of N-1, C-6 Functionalized 3,5-Dichloro-2(1H)-Pyrazinones.

Org. Biomol. Chem. 7 (2009) 2809-2815.

K. M. Orrling, M. R. Marzahn, H. Gutiérrez-de-Terán, J. Åqvist, B. M. Dunn, Mats Larhed*:

α-Substituted Norstatines as the Transition-State Mimic in Inhibitors of Multiple Digestive Vacuole Malaria Aspartic Proteases.

Bioorg. Med. Chem. 17 (2009), 5933-5949.

O. Lagerlund, M. L. H. Mantel, M. Larhed*:

Aminocarbonylations of Alkenyl Phosphates, -Chlorides, -Bromides, and -Triflates with Mo(CO)₆ as a Solid CO Source.

Tetrahedron 65 (2009), 7646-7652.

L. R. Odell, M. T. Nilsson, J. Gising, O. Lagerlund, D. Muthas, A. Nordqvist, A. Karlén, M. Larhed*:

Functionalized 3-Amino-imidazo[1,2-a]pyridines: A Novel Class of Drug-Like Mycobacterium tuberculosis Glutamine Synthetase Inhibitors.

Bioorg. Med. Chem. Lett. 19 (2009) 4790-4793.

F. Wångsell, F. Russo, J. Sävmarker, Å. Rosenquist, B. Samuelsson, M. Larhed*:

Design and synthesis of BACE-1 inhibitors utilizing a tertiary hydroxyl motif as the transition state mimic.

Bioorg. Med. Chem. Lett. 19 (2009) 4711-4714.

Book Chapters



In Handbook of Green Chemistry, Volume 1, Homogenous Catalysis, Crabtree, R. H., Anastas et al., Eds. Wiley-VCH, 2009, 79-99.

Papers: Wiki Pages

2009